N-(heterocycle-methyl)alkylamine derivative, process for producing the same, and bactericide

• US 20050101783A1
• Filed: 05/09/2001
• Published: 05/12/2005
• Est. Priority Date: 05/09/2000
• Status: Abandoned Application

• Current Assignee: Kureha Corporation
• Original Assignee: Kureha Corporation
• Inventors: Ito, Atsushi, Kusano, Nobuyuki, Araki, Nobuyuki, Sudo, Keiichi, Niizeki, Yoshitaka, Eizuka, Takayoshi, Watanabe, Tsumoru
• Application Number:
  US10/477,338
• Publication Number:
  US 20050101783A1
• Time in Patent Office: Days
• US Class Current: 546/329
• CPC Class Codes: A01N 43/36 five-membered rings
• CPC Class Codes: A01N 43/40 six-membered rings
• CPC Class Codes: A01N 43/50 1,3-Diazoles; Hydrogenated 1,3-diazoles
• CPC Class Codes: A01N 43/54 1,3-Diazines; Hydrogenated 1,3-diazines
• CPC Class Codes: A01N 43/56 1,2-Diazoles; Hydrogenated 1,2-diazoles
• CPC Class Codes: A01N 43/60 1,4-Diazines; Hydrogenated 1,4-diazines
• CPC Class Codes: A01N 43/653 1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
• CPC Class Codes: A01N 43/78 1,3-Thiazoles; Hydrogenated 1,3-thiazoles
• CPC Class Codes: A61P 31/10 Antimycotics

Abstract

A N-heterocyclicmethyl-alkylamine derivative according to the present invention is a N-heterocyclicmethyl-alkylamine derivative represented by the following general formula (I): or an acid addition salt thereof.
[in the formula, R¹ represents a heterocycle which has at least one nitrogen atom as a hetero atom and may have a substituent on a ring; R² represents a hydrogen or the like; R³ represents an alkyl group having a carbon number of 1 to 5 or the like; R⁴ represents an alkyl group having a carbon number of 1 to 5 or the like; when R⁴ is an alkyl group having a carbon number of 1 to 5 or a halogenated alkyl group having a carbon number of 1 to 5, carbon atoms in R³ and R⁴ may be bonded to form a ring structure; m represents an integer of 1 to 3; R⁵ represents a cycloalkyl group or the like described by the following formula (III):
(in the formula, Y and Z each represents a hydrogen atom or the like, the letter p represents an integer of 2 to 5, and the groups described by CYZ may be each the same or different), when m is 1 and R⁴ is a hydrogen atom, R⁵ is a cycloalkyl group described by the foregoing formula (III).]

Claims

1. A N-heterocyclicmethyl-alkylamine derivative represented by the following general formula (I) or an acid addition salt thereof:

2. A method of manufacturing a N-heterocyclicmethyl-alkylamine derivative including a process which obtains a N-heterocyclicmethyl-alkylamine derivative represented by the following formula (I):

4. The method of manufacturing the N-heterocyclicmethyl-alkylamine derivative according to claim 2, wherein the aldehyde derivative represented by the following formula (IV):

5. The method of manufacturing the N-heterocyclicmethyl-alkylamine derivative according to claim 2, wherein the aldehyde derivative represented by the following formula (IV):

6. The method of manufacturing the N-heterocyclicmethyl-alkylamine derivative according to claim 2, wherein the aldehyde derivative represented by the following formula (IV):

3. A method of manufacturing a N-heterocyclicmethyl-alkylamine derivative including a process which obtains a N-heterocyclicmethyl-alkylamine derivative represented by the following formula (I):

7. The method of manufacturing the N-heterocyclicmethyl-alkylamine derivative according to claim 3, wherein the alkylamine derivative represented by the following formula (VI):

8. The method of manufacturing the N-heterocyclicmethyl-alkylamine derivative according to claim 3, including a process which obtains the alkylamine derivative represented by the following formula (VI):

9. A fungicide containing a N-heterocyclicmethyl-alkylamine derivative represented by the following general formula (I):