Pharmaceutical compositions containing exendins
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Abstract
Methods for treating conditions or disorders which can be alleviated by reducing food intake are disclosed which comprise administration of an effective amount of an exendin or an exendin agonist, alone or in conjunction with other compounds or compositions that affect satiety. The methods are useful for treating conditions or disorders, including obesity, Type II diabetes, eating disorders, and insulin-resistance syndrome. The methods are also useful for lowering the plasma glucose level, lowering the plasma lipid level, reducing the cardiac risk, reducing the appetite, and reducing the weight of subjects. Pharmaceutical compositions for use in the methods of the invention are also disclosed.
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Citations
71 Claims
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1-31. -31. (canceled)
- 32. A pharmaceutical composition comprising an exendin-4 and a buffer, wherein said composition has a pH of from about 3.0 to about 8.0.
- 52. A pharmaceutical composition comprising exendin-4, mannitol, and an acetate buffer, wherein said composition has a pH of about 4.5.
- 56. A pharmaceutical composition comprising an exendin-3 and a buffer, wherein said composition has a pH of from about 3.0 to about 8.0.
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71. A pharmaceutical composition comprising an exendin selected from the group consisting of exendin-4 (1-30), exendin-4 (1-30) amide, exendin-4 (1-28) amide, 14Leu, 25Phe exendin-4 amide, 4Leu, 25Phe exendin-4 (1-28) amide, 14Leu, 22Ala, 25Phe exendin-4 (1-28) amide, and any combination thereof;
- and a buffer, wherein said composition has a pH of from about 3.0 to about 8.0.
Specification