QUINAZOLINONES AS INHIBITORS OF HUMAN PHOSPHATIDYLINOSITOL 3-KINASE DELTA
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Abstract
Compounds that inhibit PI3Kδ activity, including compounds that selectively inhibit PI3Kδ activity, are disclosed. Methods of inhibiting phosphatidylinositol 3-kinase delta isoform (PI3Kδ) activity, and methods of treating diseases, such as disorders of immunity and inflammation in which PI3Kδ plays a role in leukocyte function, using the compounds also are disclosed.
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Citations
44 Claims
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1-32. -32. (canceled)
- 33. A compound, wherein the compound is
- 39. A method of treating a condition in a subject, wherein the condition is cancer, comprising administering to a subject in need thereof an effective amount of a compound, wherein the compound is 6-fluoro-3-phenyl-2-[1-(9H-purin-6-ylamino)-ethyl]-3H-quinazolin-4-one or a pharmaceutically acceptable salt thereof.
Specification