FORMULATIONS OF BISPHOSPHONATES AND VITAMIN D SUIUTABLE FOR INTERMITTENT INTRAMUSCULAR AND SUBCUTANEOUS ADMINISTRATION
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Abstract
Compositions for pharmaceutical use are described, comprising bisphosphonates and vitamin D in high concentration, destined to the intramuscular and subcutaneous intermittent administration for treatment of bone and skeletal system diseases, particularly osteoporosis, and sensitive cancers. These formulations are characterized by the use of a lipid and phospholipid emulsion at high concentration, having optimal carrier and solvent power for both the pharmacologically active components.
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Citations
53 Claims
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1-24. -24. (canceled)
- 25. A composition for pharmaceutical use comprising a substance of the class of bisphosphonates and vitamin D, wherein all components are dissolved in an emulsion comprising lipids and phospholipids in water at concentration of at least 5% and 0.5% w/v respectively, and in a volume suitable for an intramuscular or subcutaneous administration.
Specification