BORONIC ACID DERIVATIVES AND THERAPEUTIC USES THEREOF
First Claim
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1. A compound having the structure of the Formula I or II, or pharmaceutically acceptable salts thereof:
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Abstract
Disclosed herein are antimicrobial compounds compositions, pharmaceutical compositions, the method of use and preparation thereof. Some embodiments relate to boronic acid derivatives and their use as therapeutic agents, for example, β-lactamase inhibitors (BLIs).
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Citations
86 Claims
- 1. A compound having the structure of the Formula I or II, or pharmaceutically acceptable salts thereof:
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37. A compound having the structure of the Formula III or IV, or pharmaceutically acceptable salts thereof:
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52. A compound having the structure of Formula V, or pharmaceutically acceptable salts thereof:
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66. A compound having the structure of Formula VI, or pharmaceutically acceptable salts thereof:
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Specification