TRIAZOLOPYRIDINES AND TRIAZOLOPYRAZINES AS LSD1 INHIBITORS
2 Assignments
0 Petitions
Accused Products
Abstract
The present invention is directed to [1,2,4]triazolo[1,5-a]pyridine and [1,2,4]triazolo[1,5-a]pyrazine derivatives which are LSD1 inhibitors useful in the treatment of diseases such as cancer.
-
Citations
79 Claims
-
1-45. -45. (canceled)
- 46. A method of treating a disease, wherein said disease is selected from leukemia, lung cancer, Ewing'"'"'s sarcoma, prostate cancer, and myelofibrosis, comprising administering to a patient a therapeutically effective amount of a compound of Formula I:
Specification