NOVEL N-(3,5-DIHALOPHENYL)-IMIDE COMPOUNDS

• US 3,745,170 A
• Filed: 03/06/1970
• Issued: 07/10/1973
• Est. Priority Date: 03/19/1969
• Status: Expired due to Term

• Current Assignee: Akiba K, Fujinami A, Kameda N, Nodera K, Ooba S, Ooishi T, Ozaki T, Tanaka K, Yamamoto S
• Original Assignee: Akiba K, Fujinami A, Kameda N, Nodera K, Ooba S, Ooishi T, Ozaki T, Tanaka K, Yamamoto S
• Inventors: FUJINAMI A, OZAKI T, KAMEDA N, AKIBA K, OOISHI T, NODERA K, TANAKA K, OOBA S, YAMAMOTO S
• Application Number:
  US05/017,339
• Time in Patent Office: 1,222 Days
• US Class Current: 548/544
• CPC Class Codes: C07D 207/40 2,5-Pyrrolidine-diones
• CPC Class Codes: C07D 207/408 Radicals containing only hydrogen and carbon atoms attached to ring carbon atoms
• CPC Class Codes: C07D 207/44 having three double bonds between ring members or between ring members and non-ring members
• CPC Class Codes: C07D 207/452 with hydrocarbon radicals, substituted by hetero atoms, directly attached to the ring nitrogen atom
• CPC Class Codes: C07D 209/48 with oxygen atoms in positions 1 and 3, e.g. phthalimide
• CPC Class Codes: C07D 209/52 condensed with a ring other than six-membered
• CPC Class Codes: C07D 211/88 attached in positions 2 and 6, e.g. glutarimide
• CPC Class Codes: C07D 295/15 to an acyclic saturated chain

Abstract

NOVEL N-(3,5-DIHOLOPHENYL)IMIDE COMPOUNDS, WHICH EXHIBIT A STRONG ANTIMICROBIAL ACTIVITY AGAINST MICROORGANISMS INCLUDING PHYTOPATHOGENIC FUNGI, PARASITES OF INDUSTRIAL PRODUCTS AND PATHOGENIC MICROORGANISMS, REPRESENTED BY THE FORMULA,

(3-X,5-X'"'"''"'"'-PHENYL)-N<(-CO-A-CO-)

WHEREIN X AND X'"'"''"'"' EACH REPRESENT HALOGENS AND A REPRESENTS A SUBSTITUTED ETHYLENE SUCH AS CHLOROETHYLENE, C1C4 ALKYLTHIOETHYLENE, C1-C2 ALKYL-ETHYLENE OR 1,2-DI-C1C2-ALKYL-ETHYLENE, A CYCLOPROPYLENE SUCH AS 1,3-DIMETHYLCYCLOPROPYLENE, TRIMETHYLENE, A CYCLOHEXYLENE-1,2-, CYCLOHEXENYLENE-1,2-, CYCLOHEXADIENYLENE-1,2- OR O-PHENYLENE. THE N-(3,5-DIHALOPHENY)IMIDE COMPOUNDS CAN BE OBTAINED BY ANY OF METHODS WHICH PRODUCE IMIDE COMPOUNDS ON REACTION OF AN N-(3,5-DIHALOPHENYL)MALEIMIDE COMPOUND WITH A MERCAPTAN, A HYDROGEN HALIDE, PHOSPHORUS CHLORIDE OR THIONYLCHLORIDE.

Claims