Fucosidase inhibitor
First Claim
Patent Images
1. A method for the production of 2,6-imino-2,6,7-trideoxy-D-glycero-D-gluco-heptitol comprising catalytically hydrogenating 6-azido-7-O-tert-butyldimethylsilyl-1,6-dideoxy-3,4-O-isopropylidene-L-gulo-heptulo -2-ose with platinum (IV) oxide at about room temperature followed by hydrolytic removal of the silyl and isopropylidene protecting groups.
0 Assignments
0 Petitions
Accused Products
Abstract
The synthesis of the novel fucosidase inhibitor, 2,6-imino-2,6,7-trideoxy-D-glycero-D-gluco heptitol, is disclosed.
-
Citations
2 Claims
- 1. A method for the production of 2,6-imino-2,6,7-trideoxy-D-glycero-D-gluco-heptitol comprising catalytically hydrogenating 6-azido-7-O-tert-butyldimethylsilyl-1,6-dideoxy-3,4-O-isopropylidene-L-gulo-heptulo -2-ose with platinum (IV) oxide at about room temperature followed by hydrolytic removal of the silyl and isopropylidene protecting groups.
Specification