Heterocyclic analgesic compounds and methods of use thereof
First Claim
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1. A compound represented by G:
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wherein R represents phenyl, 2-fluorophenyl, 3-fluorophenyl, or 4-fluorophenyl;
R′
represents H or OH; and
the stereochemical configuration at any stereocenter of a compound represented by G is R, S, or a mixture of these configurations.
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Abstract
One aspect of the present invention relates to novel heterocyclic compounds. A second aspect of the present invention relates to the use of the novel heterocyclic compounds as ligands for various cellular receptors, including opiate receptors, other G-protein-coupled receptors, and ion channels. An additional aspect of the present invention relates to the use of the novel heterocyclic compounds as analgesics.
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26 Claims
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1. A compound represented by G:
-
wherein R represents phenyl, 2-fluorophenyl, 3-fluorophenyl, or 4-fluorophenyl;
R′
represents H or OH; and
the stereochemical configuration at any stereocenter of a compound represented by G is R, S, or a mixture of these configurations. - View Dependent Claims (2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 19, 20, 21, 22, 23, 24, 25, 26)
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Specification