Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors
First Claim
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1. A method of inhibiting an activity of JAK2 comprising contacting said JAK2 with a compound of Formula I:
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Abstract
The present invention provides pyrrolo[2,3-b]pyridine-4-yl amines pyrrolo[2,3-b]pyrimidin-4-yl amines that modulate the activity of Janus kinases and are useful in the treatment of diseases related to activity of Janus kinases including, for example, immune-related diseases and cancer.
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9 Claims
- 1. A method of inhibiting an activity of JAK2 comprising contacting said JAK2 with a compound of Formula I:
- 3. A method of treating a skin disorder in a patient comprising topically administering to said patient a therapeutically effective amount of a compound of Formula II:
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