Dosage and formulation
First Claim
1. A pharmaceutical composition comprising aclidinium in the form of a dry powder of a pharmaceutically acceptable salt in admixture with a pharmaceutically acceptable dry powder carrier, wherein the pharmaceutical composition is in a dosage form which provides a) a metered nominal dose of aclidinium equivalent to 200 micrograms aclidinium bromide (plus/minus 35%), b) an emitted dose of aclidinium equivalent to 180 micrograms (plus/minus 35%) aclidinium bromide, or c) a fine particle dose of aclidinium equivalent to 60 micrograms (plus/minus 35%) aclidinium bromide, wherein the pharmaceutical composition is for inhalation.
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Accused Products
Abstract
The present disclosure relates to pharmaceutical compositions for inhalation comprising aclidinium in the form of a dry powder of a pharmaceutically acceptable salt in admixture with a pharmaceutically acceptable dry powder carrier, providing a metered nominal dose of aclidinium equivalent to about 200 micrograms aclidinium bromide.
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Citations
23 Claims
- 1. A pharmaceutical composition comprising aclidinium in the form of a dry powder of a pharmaceutically acceptable salt in admixture with a pharmaceutically acceptable dry powder carrier, wherein the pharmaceutical composition is in a dosage form which provides a) a metered nominal dose of aclidinium equivalent to 200 micrograms aclidinium bromide (plus/minus 35%), b) an emitted dose of aclidinium equivalent to 180 micrograms (plus/minus 35%) aclidinium bromide, or c) a fine particle dose of aclidinium equivalent to 60 micrograms (plus/minus 35%) aclidinium bromide, wherein the pharmaceutical composition is for inhalation.
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14. A method of treating a respiratory condition chosen from asthma and chronic obstructive pulmonary disease, comprising administering a pharmaceutical composition comprising aclidinium in the form of a dry powder of a pharmaceutically acceptable salt in admixture with a pharmaceutically acceptable dry powder carrier, wherein the pharmaceutical composition is in a dosage form which provides:
- a) a metered nominal dose of aclidinium equivalent to 200 micrograms (plus/minus 35%) aclidinium bromide, b) an emitted dose of aclidinium equivalent to 180 micrograms (plus/minus 35%) aclidinium bromide, or c) a fine particle dose of aclidinium equivalent to 60 micrograms (plus/minus 35%) aclidinium bromide, by inhalation to a patient in need of such treatment.
- View Dependent Claims (15, 16, 17, 18, 20, 21)
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19. A multidose dry powder inhaler device comprising a pharmaceutical composition comprising aclidinium in the form of a dry powder of a pharmaceutically acceptable salt in admixture with a pharmaceutically acceptable dry powder carrier, wherein the pharmaceutical composition is in a dosage form which provides, and the device is calibrated to deliver upon actuation:
- a) a metered nominal dose of aclidinium equivalent to 200 micrograms (plus/minus 35%) of aclidinium bromide, b) an emitted dose of aclidinium equivalent to 180 micrograms (plus/minus 35%) aclidinium bromide, or c) a fine particle dose of aclidinium equivalent to 60 micrograms (plus/minus 35%) aclidinium bromide.
Specification