Substituted pyrrolo[2,3-b]pyridines for treating cancer or inflammatory diseases
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Abstract
Disclosed herein are substituted pyrrolopyridine and pyrrolopyrazine compounds and compositions useful in the treatment of TAK mediated diseases, such as cancer, having the structure of Formula (I):
wherein R1, R2, R3, and R4 are as defined in the detailed description. Methods of modulation of TAK activity in a human or animal subject are also provided, providing therapeutic benefit to subjects with disease conditions, especially cancer.
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Citations
10 Claims
- 1. A compound of Formula (I):
- 8. A compound selected from the group consisting of:
Specification