Processes for preparing isoquinolinones and solid forms of isoquinolinones
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Abstract
Polymorphs of chemical compounds that modulate kinase activity, including PI3 kinase activity, and compounds, pharmaceutical compositions, and methods of treatment of diseases and conditions associated with kinase activity, including P13 kinase activity, are described herein. Also provided herein are processes for preparing compounds, polymorphs thereof, and pharmaceutical compositions thereof.
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Citations
66 Claims
- 1. A compound of Formula (I):
- 2. A mixture of two or more compounds of Formula (I):
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3. A mixture of two or more compounds of Formula (I):
- 5. Polymorph Form C of a compound of Formula (I):
- 9. Polymorph Form B of a compound of Formula (I):
- 13. Polymorph Form D of a compound of Formula (I):
- 17. Polymorph Form E of a compound of Formula (I):
- 21. Polymorph Form F of a compound of Formula (I):
- 25. Polymorph Form G of a compound of Formula (I):
- 29. Polymorph Form H of a compound of Formula (I):
- 33. Polymorph Form I of a compound of Formula (I):
- 37. Polymorph Form J of a compound of Formula (I):
- 42. A pharmaceutical composition comprising a therapeutically effective amount of a compound of Formula (I):
- 47. Polymorph Form A of a compound of Formula (I):
Specification