Substituted aminoquinazolone (thio-ketone) derivative or its salt, its intermediate and pest controlling agent and its application method

Substituted aminoquinazolone (thio-ketone) derivative or its salt, its intermediate and pest controlling agent and its application method

  • CN 1,302,801 A
  • Filed: 11/02/2000
  • Published: 07/11/2001
  • Est. Priority Date: 11/02/1999
  • Status: Abandoned Application
First Claim
Patent Images

1. aminoquinazolinone (thioketones) derivative of the replacement of general formula (I) expression, or its salt:

  • Wherein R is hydrogen atom;

    Hydroxyl;

    Formoxyl;

    (C1- 12) alkyl;

    Halo (C1-6) alkyl;

    Hydroxyl (C1-6) alkyl;

    (C2-6) alkenyl;

    (C2-6) alkynyl;

    (C1-6) alkoxyl;

    Halo (C1-6) alkoxyl;

    (C1-6) alkoxyl (C1-3) alkyl;

    (C1-6) alkoxyl (C1-3) alkoxyl (C1-3) alkyl;

    (C1-6) alkylthio group;

    Halo (C1-6) alkylthio group;

    (C1-6) the alkyl sulfinyl;

    (C1-6) the alkyl sulfonyl base;

    (C1-6) alkylthio group (C1-3) alkyl;

    Two (C1-6) alkoxyl (C1-3) alkyl, wherein (C1-6) alkoxyl can be identical or different;

    Unsubstituted amino (C1-6) alkyl;

    Has the amino (C of one or two substituent replacement1-6) alkyl, wherein substituting group can be identical or different, is selected from (C1-6) alkyl, halo (C1-6) alkyl, (C2-6) alkenyl and (C2-6) alkynyl;

    Cyano group (C1-6) alkyl;

    (C1-6) the alkyl carbonyl;

    (C1-6) the alkoxyl carbonyl;

    Hydroxyl carbonyl (C1-3) alkyl;

    (C1-6) alkoxyl carbonyl (C1-3) alkyl;

    Unsubstituted amino carbonyl;

    Have one or two substituent substituted aminocarbonyl, wherein substituting group can be identical or different, is selected from (C1-6) alkyl, (C2-6) alkenyl and (C2-6) alkynyl;

    (C3-6) cycloalkyl (C1-3) alkyl;

    Unsubstituted phenyl (C1-3) alkyl;

    Have 1-5 substituent replacement phenyl (C on ring1-3) alkyl, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1- 6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group and halo (C1-6) alkylthio group;

    Unsubstituted phenylcarbonyl group;

    Have 1-5 substituent replacement phenylcarbonyl group on ring, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group and halo (C1-6) alkylthio group;

    Unsubstituted thiophenyl;

    Have 1-5 substituent substituted benzene sulfenyl on ring, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group and halo (C1-6) alkylthio group;

    Unsubstituted phenyl sulfonyl;

    Have 1-5 substituent substituted phenyl sulfonyl base on ring, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group and halo (C1-6) alkylthio group;

    Unsubstituted phenyl (C1-6) the alkyl sulfonyl base;

    Have 1-5 substituent replacement phenyl (C on ring1-6) the alkyl sulfonyl base, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group and halo (C1-6) alkylthio group;

    Unsubstituted phenyloxycarbonyl;

    Have 1-5 substituent substituent phenoxy carbonyl on ring, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group and halo (C1-6) alkylthio group;

    Unsubstituted phenoxy group (C1-3) alkyl;

    Have 1-5 substituent substituent phenoxy (C on ring1-3) alkyl, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group and halo (C1-6) alkylthio group;

    Unsubstituted phenyl (C2-6) alkenyl;

    Have 1-5 substituent replacement phenyl (C on ring2-6) alkenyl, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group, halo (C1-6) alkylthio group and (C1-2) alkylenedioxy group;

    Unsubstituted phenyl (C2-6) alkynyl;

    Have 1-5 substituent replacement phenyl (C on ring2-6) alkynyl, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group, halo (C1-6) alkylthio group and (C1-2) alkylenedioxy group;

    Unsubstituted phenyl (C2-4) alkynyl (C1-3) alkyl;

    Have 1-5 substituent replacement phenyl (C on ring2-4) alkynyl (C1-3) alkyl, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxyl, halo (C1-6) alkoxyl, (C1-6) alkylthio group halo (C1-6) alkylthio group and (C1-2) alkylenedioxy group;

    DOX-2-base (C1-3) alkyl;

    Or phthaloyl imino (C1-6) alkyl,R 1Be to have 1-3 heteroatomic 5-or 6-unit heterocycle, wherein heteroatoms can be identical or different, is selected from Sauerstoffatom, and sulphur atom and nitrogen-atoms, described heterocycle can have 1-5 substituting group, and wherein substituting group can be identical or different, is selected from halogen atom, cyano group, (C 1-6) alkyl, halo (C 1-6) alkyl and (C 1-6) alkoxyl group, and assorted ring nitrogen can form the N-oxide groups, Y is Sauerstoffatom or sulphur atom,Z is-N=C (R 2)-(be R wherein 2Be hydrogen atom, (C 1-6) alkyl or halo (C 1-6) alkyl), or -N (R 3)-CH (R 2)-(be R wherein 2Define as above, and R 3Be hydrogen atom, (C 1-6) alkyl, formyl radical, (C 1-3) alkyl-carbonyl or halo (C 1-3) the alkyl base), X can be identical or different, is bromine atoms, the iodine atom;

    Hydroxyl;

    Cyano group;

    (C 1-6) alkyl;

    Halo (C 1-10) alkyl;

    (C 2-5) alkenyl;

    Halo (C 2-6) alkenyl;

    (C 2-6) alkynyl;

    (C 1-6) alkoxyl group;

    Halo (C 1-6) alkoxyl group;

    (C 1-6) alkylthio;

    Halo (C 1-6) alkylthio;

    (C 1-6) alkyl sulphinyl;

    Halo (C 1-6) alkyl sulphinyl;

    (C 1-6) alkyl sulphonyl;

    Halo (C 1-6) alkyl sulphonyl;

    Halo (C 1-6) halogenated alkoxy (C 1-6) alkoxyl group;

    Carboxyl;

    (C 1-6) carbalkoxy;

    Unsubstituted aminocarboxyl;

    Have one or two substituent substituted aminocarbonyl, wherein substituting group can be identical or different, is selected from (C 1-6) alkyl, (C 2-6) alkenyl and (C 2-6) alkynyl;

    Carboxyl (C 1-6) alkyl;

    (C 1-6) carbalkoxy (C 1-3) alkyl;

    Unsubstituted aminocarboxyl (C 1-3) alkyl;

    Has one or two substituent substituted aminocarbonyl (C 1-3) alkyl, wherein substituting group can be identical or different, is selected from (C 1-6) alkyl, (C 2-6) alkenyl and (C 2-6) alkynyl;

    Sulfonic group;

    Unsubstituted amino-sulfonyl;

    (C 1-6) the alkoxyl group alkylsulfonyl;

    Have one or two substituent substituted-amino alkylsulfonyl, wherein substituting group can be identical or different, is selected from (C 1-6) alkyl, (C 2-6) alkenyl and (C 2-6) alkynyl;

    Unsubstituted phenyl;

    Have 1-5 substituent substituted-phenyl on the ring, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C 1-6) alkyl, halo (C 1-6) alkyl, (C 1-6) alkoxyl group, halo (C 1-6) alkoxyl group, (C 1-6) alkylthio, halo (C 1-6) alkylthio, (C 1-6) alkoxyl group alkylsulfonyl and have one or two substituent substituted-amino alkylsulfonyl, wherein substituting group can be identical or different, is selected from (C 1-6) alkyl, (C 2-6) alkenyl and (C 2-6) alkynyl;

    Unsubstituted phenyl (C 1-3) alkyl;

    Have 1-5 substituent substituted-phenyl (C on the ring 1-3) alkyl, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C 1-6) alkyl, halo (C 1-6) alkyl, (C 1-6) alkoxyl group, halo (C 1-6) alkoxyl group, (C 1-6) alkylthio and halo (C 1-6) alkylthio;

    Unsubstituted phenoxy;

    Have 1-5 substituent substituent phenoxy on the ring, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C 1-6) alkyl, halo (C 1-6) alkyl, (C 1-6) alkoxyl group, halo (C 1-6) alkoxyl group, (C 1-6) alkylthio and halo (C 1-6) alkylthio;

    Unsubstituted pyridine oxygen base;

    Have one or more substituent substituted pyridines oxygen bases on the ring, wherein substituting group can be identical or different, is selected from halogen atom, nitro, cyano group, (C 1-6) alkyl, halo (C 1-6) alkyl, (C 1-6) alkoxyl group, halo (C 1-6) alkoxyl group, (C 1-6) alkylthio and halo (C 1-6) alkylthio;

    And n is 0 to 4 integer.

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